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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T11486 | GSK2807 Trifluoroacetate | Histone Methyltransferase | |
GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM). | |||
T69738 | GSK-2807 free base | ||
GSK2807 is a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM). GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3. GSK2807 may be useful for cancer trea... |